Target List
Neurotransmitter Receptors
Adenosine Receptors
ADORA1, ADORA2A, ADORA2B, ADORA3
Adrenergic Receptors
ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3
Cannabinoid Receptors
CNR1, CNR2
Dopamine Receptors
DRD1, DRD2, DRD3, DRD4, DRD5
Gamma-Aminobutyric Acid (GABA) Receptors
GABBR1, GABBR2
Muscarinic Cholinergic Receptors
CHRM1, CHRM2, CHRM3, CHRM4, CHRM5
Opioid Receptors
OGFR, OPRD1, OPRK1, OPRL1, OPRM1
Ionotropic Glutamate Receptors
GRIK3
Metabotropic Glutamate Receptors
GRM1, GRM2, GRM3, GRM4, GRM5, GRM6, GRM7, GRM8
Serotonin (5-Hydroxytryptamine) Receptors
HTR1A, HTR1B, HTR1D, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR3A, HTR3B, HTR4, HTR5A, HTR6, HTR7
Neuropeptide Receptors
Galanin Receptors
GALR1, GALR2, GALR3
Hypocretin (Orexin) Receptors
HCRTR1, HCRTR2
Neuromedin Receptors
NMBR, NMUR1, NMUR2
Neuropeptide Receptors
NPBWR1, NPBWR2, NPFFR1, NPFFR2, NPSR1, NPY1R, NPY2R, NPY5R
Neurotensin Receptors
NTSR1, NTSR2
Tachykinin Receptors
TACR1, TACR2, TACR3
Hormone Receptors
Calcitonin Receptors
CALCR, CALCRL
Cholecystokinin Receptors
CCKAR, CCKBR
Corticotropin Releasing Hormone Receptors
CRHR1, CRHR2
Glucagon-Like Peptide Receptors
GLP1R, GLP2R
Melanin-Concentrating Hormone Receptors
MCHR1, MCHR2
Melanocortin Receptors
MC1R, MC2R, MC3R, MC4R, MC5R
Parathyroid Hormone Receptors
PTH1R, PTH2R
Prokineticin Receptors
PROKR1, PROKR2
Somatostatin Receptors
SSTR1, SSTR2, SSTR3, SSTR4, SSTR5
Other Hormone Receptors
APLNR, ADGRE1 (EMR1), FSHR, GCGR, GHRHR, GHSR, GIPR, GNRHR, GRPR, LEPR, LHCGR, PRLHR, SCTR, TRHR, TSHR
Orphan G-Protein Coupled Receptors (GPCRs)
GPR1, GPR101, ADGRF1, ADGRF2, ADGRG4, ADGRF3, ADGRG5, ADGRF4, ADGRF5, GPR119, GPR12, FFAR4, ADGRA1, ADGRA2, ADGRA3, ADGRG6, ADGRG7, GPR132, ADGRD1, GPR135, GPR139, GPR141, GPR142, GPR143, ADGRD2, GPR146, GPR148, GPR149, GPR15, GPR150, GPR151, GPR152, GPR153, GPR156, GPR157, GPR158, GPR160, GPR161, GPR162, GPR17, GPR171, GPR173, GPR174, GPR176, GPR179, GPR18, GPR182, GPR183, GPR19, GPR20, GPR21, GPR22, GPR25, GPR26, GPR27, GPR3, GPR31, GPR32, GPR34, GPR35, GPR37, GPR37L1, GPR39, GPR4, PTGDR2 (CRTH2, GPR44), GPR45, GPR50, GPR52, GPR55, ADGRG1, GPR6, GPR61, GPR62, GPR63, ADGRG2, GPR65, GPR68, GPR75, C5AR2, GPR78, HCAR1, GPR82, GPR83, GPR84, GPR85, GPR87, GPR88, ADGRG3, ADGRV1, GPRC5A, GPRC5B, GPRC5C, GPRC5D, GPRC6A
Angiogenesis & Vasoactivity
Angiotensin II Receptors
AGTR1, AGTR2
Arginine Vasopressin Receptors
AVPR1A, AVPR1B, AVPR2
Bradykinin Receptors
BDKRB1, BDKRB2
Brain-Specific Angiogenesis Inhibitors
ADGRB1 (BAI1), ADGRB2, ADGRB3
Endothelin Receptors
EDNRA, EDNRB
Natriuretic Peptide Receptors
NPR1, NPR2, NPR3
Vasoactive Intestinal Peptide Receptors
VIPR1, VIPR2
Inflammation & Immune System Regulation
Complement Component Receptors
C3AR1, C5AR1 (GPR77)
Chemokine & Cytokine Receptors
ACKR2, CCR1, CCR10, CCR2, CCR3, CCR4, CCR5, CCR6, CCR7, CCR8, CCR9, ACKR4, CCRL2, CMKLR1, CX3CR1, CXCR3, CXCR4, CXCR5, CXCR6, ACKR3, CXCR1, CXCR2, XCR1 (CCXCR1)
Histamine Receptors
HRH1, HRH2, HRH3, HRH4
Lipid Messenger Receptors
Cysteinyl Leukotriene Receptors
CYSLTR1, CYSLTR2
Free Fatty Acid Receptors
FFAR1, FFAR2, FFAR3
Leukotriene B4 & Thromboxane Receptors
LTB4R, LTB4R2, TBXA2R
Lysophosphatidic Acid Receptors
LPAR1, LPAR2, LPAR3, LPAR4, LPAR5
Prostaglandin Receptors
PTGDR, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR
Sphingosine-1-Phosphate Receptors
S1PR1, S1PR2, S1PR3, S1PR4, S1PR5
Growth Factor Receptors
Frizzled Homologs
FZD1, FZD10, FZD2, FZD3, FZD4, FZD5, FZD6, FZD7, FZD8, FZD9
Platelet-Derived Growth Factor Receptors
PDGFRB, PDGFRL
Other G-Protein Coupled Receptors (GPCRs)
Coagulation Factor II (Thrombin) Receptors
F2R (PAR1), F2RL1 (PAR2), F2RL2 (PAR3), F2RL3 (PAR4)
Cadherin, EGF LAG Seven-Pass G-Type Receptors (Flamingo Homologs)
CELSR1, CELSR2, CELSR3
Formyl Peptide Receptors
FPR1, FPR2, FPR3
Leucine-Rich Repeat-Containing G-Protein Coupled Receptors
LGR4, LGR5
Latrophilins
ADGRL1, ADGRL2, ADGRL3
MAS-Related G-Protein Couple Receptors
MAS1, MRGPRD, MRGPRE, MRGPRF, MRGPRG, MRGPRX1, MRGPRX2, MRGPRX3, MRGPRX4
Melatonin Receptors
MTNR1A, MTNR1B
Opsins & Rhodopsin
OPN1SW, OPN3, OPN4, OPN5, RHO
Purinergic (P2Y) Receptors
P2RY1, P2RY10, P2RY11, P2RY12, P2RY13, P2RY14, P2RY2, P2RY4, LPAR6, P2RY6, P2RY8
Relaxin / Insulin-Like Family Peptide Receptors
RXFP1, RXFP2, RXFP3, RXFP4
Sortilin-Related VPS10 Domain Containing Receptors
SORCS1, SORCS2, SORCS3
Trace Amine Associated Receptors
TAAR1, TAAR2, TAAR5, TAAR6, TAAR9
Other G-Protein Coupled Receptors (GPCRs)
ADCYAP1R1, BRS3, CASR, ADGRE5 (CD97), CRCP, ACKR1, ADGRL4, GPBAR1, GPER1, HCAR2, KISS1R, OXGR1, OXTR, NPY4R, PTAFR, QRFPR, RGR, RRH, SIGMAR1, SMO, SUCNR1, TM2D1, UTS2R, XPR1